SCHEMBL7401437

SCHEMBL7401437

NC(=O)CC(CS)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
PKM P14618 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
ALDH1A1 P00352 1/20 0.53
GABBR2 O75899 1/20 0.52
GABBR1 Q9UBS5 1/20 0.52
CYP2C19 P33261 3/20 0.49
SLC6A3 Q01959 3/20 0.44
DRD3 P35462 2/20 0.44
LMNA P02545 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
EDNRB P24530 1/20 0.44
MAPK1 P28482 1/20 0.44
MC4R P32245 1/20 0.44
MC3R P41968 1/20 0.44
DRD2 P14416 1/20 0.44
ANPEP P15144 1/20 0.42
ENPEP Q07075 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9105247 0.88 ALDH1A1 (0.63) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL4177024 0.84 GABBR2 (0.66) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL27814502 0.82 GABBR2 (0.69) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL1059563 0.82 CYP2D6 (0.56) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL27691658 0.82 GABBR2 (0.75) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL8187229 0.82 CYP2D6 (0.56) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL8192677 0.82 CYP2D6 (0.56) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL186239 0.81 ALDH1A1 (0.56) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL186231 0.81 ALDH1A1 (0.56) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1
SCHEMBL186417 0.81 ALDH1A1 (0.56) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0280627-B1 DERIVATIVES OF N-SUBSTITUTED ALPHA-MERCAPTOMETHYL-BENZENE-PROPANAMIDE, PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICINES AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-04-21 EP disclosed
EP-0280627-B1 DERIVATIVES OF N-SUBSTITUTED ALPHA-MERCAPTOMETHYL-BENZENE-PROPANAMIDE, PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICINES AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-04-21 EP disclosed
EP-0280627-A2 Derivatives of N-substituted alpha-mercaptomethyl-benzene-propanamide, process for their preparation, their use as medicines and compositions containing them ROUSSEL-UCLAF (FR) 1988-08-31 EP disclosed
EP-0280627-A2 Derivatives of N-substituted alpha-mercaptomethyl-benzene-propanamide, process for their preparation, their use as medicines and compositions containing them ROUSSEL-UCLAF (FR) 1988-08-31 EP disclosed