SCHEMBL7401464

SCHEMBL7401464

COc1cc(C(=O)OC(C)(C)C)ccc1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA4 P22748 2/20 0.49
CA6 P23280 2/20 0.49
CA7 P43166 2/20 0.49
CA9 Q16790 2/20 0.49
CA14 Q9ULX7 2/20 0.49
TPMT P51580 1/20 0.49
HTT P42858 3/20 0.46
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45
GABRA1 P14867 1/20 0.45
GABRG2 P18507 1/20 0.45
GABRB3 P28472 1/20 0.45
GABRA3 P34903 1/20 0.45
GABRA2 P47869 1/20 0.45
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25278897 0.88 CA12 (0.49) ALDH1A1CA12CA1CA2CA4
SCHEMBL7399022 0.88 MAPT (0.50) ALDH1A1HTTKDM4EHPGDGABRA1
SCHEMBL30457729 0.88 CA12 (0.49) ALDH1A1CA12CA1CA2CA4
SCHEMBL2191714 0.86 SLC7A5 (0.43) ALDH1A1CA12CA1CA2CA4
SCHEMBL12540431 0.85 GABRA1 (0.43) CA12CA1CA2CA4CA6
SCHEMBL11238694 0.83 TSHR (0.61) ALDH1A1CA12CA1CA2CA4
SCHEMBL644612 0.83 MAPT (0.60) ALDH1A1CA12CA1CA2CA4
SCHEMBL9030031 0.82 PTPN11 (0.41) MAPT
SCHEMBL17864530 0.82 RXRB (0.47) ALDH1A1CA12CA1CA2CA9
Vanillic Acid SCHEMBL6508773 0.82 HTT (0.73) CA12CA1CA2CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714299-B1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2002-04-24 EP disclosed
US-5665719-A Benzoxazinone and benzopyrimidinone piperidinyl tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 1997-09-09 US disclosed
EP-0714299-A4 1996-07-10 EP disclosed
EP-0714299-A1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO. INC. (US) 1996-06-05 EP disclosed
WO-1995002405-A1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1995-01-26 WO disclosed