SCHEMBL740197

SCHEMBL740197

CC(C)(C)OC(=O)C1(N)CCCCC1NC(=O)c1cc2cc(Cl)ccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.51
PYGL P06737 16/20 0.48
CYP51A1 Q16850 1/20 0.46
PYGM P11217 6/20 0.45
EHMT2 Q96KQ7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL742116 0.85 SMYD3 (0.47) SMYD3PYGLPYGMEHMT2
SCHEMBL743187 0.83 F10 (0.46) SMYD3PYGLCYP51A1EHMT2
SCHEMBL741602 0.82 F10 (0.46) SMYD3PYGLCYP51A1
SCHEMBL743656 0.80 F10 (0.56)
SCHEMBL743192 0.80 F10 (0.46) SMYD3PYGLCYP51A1
SCHEMBL739574 0.79 F10 (0.45) SMYD3PYGLCYP51A1PYGM
SCHEMBL4095868 0.78 SMYD3 (0.54) SMYD3PYGLEHMT2
SCHEMBL3335058 0.78 SMYD3 (0.54) SMYD3PYGLEHMT2
SCHEMBL4083427 0.78 SMYD3 (0.54) SMYD3PYGLEHMT2
SCHEMBL3335060 0.78 SMYD3 (0.54) SMYD3PYGLEHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431370-B1 Monoacylated 1,2-diaminocycloalkanes DAIICHI SANKYO CO LTD (JP) 2013-06-19 EP disclosed
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed
US-7935824-B2 Ethylenediamine derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2011-05-03 US disclosed
EP-1270557-A1 ETHYLENEDIAMINE DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-01-02 EP disclosed