SCHEMBL7402155

SCHEMBL7402155

CCCCN1CCC(CC2CCc3cncc(C(=O)O)c3O2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 8/20 0.38
CHRM1 P11229 2/20 0.37
ADRA2B P18089 2/20 0.37
ADRA1A P35348 2/20 0.37
ADRA1B P35368 2/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
HTR1A P08908 1/20 0.37
CHRM5 P08912 1/20 0.37
ADRA2A P08913 1/20 0.37
DRD2 P14416 1/20 0.37
CHRM3 P20309 1/20 0.37
DRD4 P21917 1/20 0.37
ADRA1D P25100 1/20 0.37
HRH1 P35367 1/20 0.37
HTR2C P28335 2/20 0.36
ADRA2C P18825 1/20 0.36
HTR1D P28221 1/20 0.36
HTR2B P41595 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7411902 0.85 HTR4 (0.46) HTR4CHRM1ADRA2BADRA1AADRA1B
SCHEMBL7392357 0.79 HTR4 (0.38) HTR4CHRM1ADRA2BADRA1AADRA1B
Hydrochloric Acid SCHEMBL7417007 0.77 HTR4 (0.46) HTR4CHRM1ADRA2BADRA1AADRA1B
Hydrochloric Acid SCHEMBL7248497 0.75 HTR3A (0.53) HTR4ADRA2BADRA1AADRA1BCHRM2
SCHEMBL7401627 0.71 HTR4 (0.56) HTR4CHRM1ADRA2BADRA1AADRA1B
SCHEMBL7391971 0.71 HTR4 (0.45) HTR4CHRM1ADRA2BADRA1AADRA1B
SCHEMBL4151143 0.71 HTR4 (0.46) HTR4CHRM1ADRA2BADRA1AADRA1B
SCHEMBL7405651 0.70 HTR4 (0.55) HTR4CHRM1ADRA2BADRA1AADRA1B
SCHEMBL7399775 0.70 HTR4 (0.40) HTR4ADRA2BADRA1AADRA1BCHRM2
SCHEMBL7360909 0.70 HTR4 (0.52) HTR4ADRA2BADRA1AADRA1BCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007859-A1 5-HT4 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-04-14 WO claimed
EP-0662959-A1 5-HT4 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-07-19 EP disclosed
WO-1994007859-A1 5-HT4 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-04-14 WO disclosed