SCHEMBL7403149

SCHEMBL7403149

NC(=CC(CCc1ccccc1)C(=O)C(Cc1ccccc1)NC(=O)N1CCOCC1)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSS P25774 12/20 0.60
CTSL P07711 7/20 0.57
CTSB P07858 6/20 0.54
CTSK P43235 2/20 0.46
CTSH P09668 1/20 0.46
CTSC P53634 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7356041 0.82 CTSL (0.59) CTSSCTSLCTSBCTSKCTSH
SCHEMBL7408631 0.79 CTSS (0.61) CTSSCTSLCTSBPOLB
SCHEMBL7404835 0.79 CTSS (0.61) CTSSCTSLCTSBPOLB
SCHEMBL7354956 0.77 CTSS (0.61) CTSSCTSLCTSBCTSKCTSH
SCHEMBL7354953 0.77 CTSS (0.61) CTSSCTSLCTSBCTSKCTSH
SCHEMBL7411947 0.77 CTSS (0.58) CTSSCTSLCTSBCTSKCTSH
SCHEMBL25004070 0.77 CTSS (0.61) CTSSCTSLCTSBPOLB
SCHEMBL7275964 0.76 POLB (0.74) CTSSCTSLCTSBPOLB
SCHEMBL5193787 0.76 POLB (0.74) CTSSCTSLCTSBPOLB
SCHEMBL7354034 0.76 CTSL (0.83) CTSSCTSLCTSBCTSKCTSH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0756625-A4 IRREVERSIBLE CYSTEINE PROTEASE INHIBITORS CONTAINING VINYL GROUPS CONJUGATED TO ELECTRON WITHDRAWING GROUPS ARRIS PHARM CORP (US) 1999-07-28 EP disclosed
EP-0756625-A1 IRREVERSIBLE CYSTEINE PROTEASE INHIBITORS CONTAINING VINYL GROUPS CONJUGATED TO ELECTRON WITHDRAWING GROUPS ARRIS PHARMACEUTICAL CORPORATION (US) 1997-02-05 EP disclosed
WO-1995023222-A1 IRREVERSIBLE CYSTEINE PROTEASE INHIBITORS CONTAINING VINYL GROUPS CONJUGATED TO ELECTRON WITHDRAWING GROUPS KHEPRI PHARMACEUTICALS, INC. (US) 1995-08-31 WO disclosed