SCHEMBL7404113

SCHEMBL7404113

N#Cc1ccc2nc(Cc3nc4ccccc4[nH]3)n(CCN)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCARB1 Q8WTV0 1/20 0.46
GRIN1 Q05586 1/20 0.45
GRIN2B Q13224 1/20 0.45
TPH1 P17752 4/20 0.43
TPH2 Q8IWU9 4/20 0.43
EGFR P00533 1/20 0.42
F2 P00734 1/20 0.40
F10 P00742 1/20 0.40
F7 P08709 1/20 0.40
GAA P10253 2/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ACSS2 Q9NR19 1/20 0.39
PKM P14618 2/20 0.38
DRD4 P21917 1/20 0.37
KDM4E B2RXH2 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400871 0.84 TPH1 (0.43) SCARB1GRIN1GRIN2BTPH1TPH2
SCHEMBL7407177 0.80 F10 (0.64) F2F10F7
SCHEMBL7407685 0.80 F10 (0.48) TPH1TPH2F2F10F7
SCHEMBL7407680 0.78 F10 (0.49) TPH1TPH2F2F10F7
SCHEMBL7405159 0.72 F10 (0.55) F2F10F7
SCHEMBL7265526 0.70 GAA (0.69) GRIN1GRIN2BEGFRGAAHPGD
SCHEMBL7408187 0.69 F10 (0.58) F2F10F7GAA
SCHEMBL7407441 0.68 F10 (0.57) F2F10F7
SCHEMBL7655135 0.68 RAD52 (0.61) GRIN1GRIN2BALDH1A1MAPTPKM
SCHEMBL1638406 0.68 ACSS2 (0.43) MAPTHPGDACSS2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999026932-A1 BY AMIDINO GROUP SUBSTITUTED HETEROCYCLIC DERIVATIVES AND THEIR USE AS ANTICOAGULANTS AXYS PHARMACEUTICALS, INC. (US) 1999-06-03 WO disclosed