SCHEMBL7405189

SCHEMBL7405189

CC(C)(C)OC(=O)CCC(NC(=O)C1(C(=O)NC(C=O)CC(=O)OC(C)(C)C)CC1)C(=O)Nc1cccc(Oc2ccccc2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.40
HDAC4 P56524 4/20 0.40
HDAC2 Q92769 5/20 0.39
HDAC8 Q9BY41 4/20 0.39
HDAC3 O15379 3/20 0.39
HDAC7 Q8WUI4 3/20 0.39
HDAC10 Q969S8 3/20 0.39
HDAC11 Q96DB2 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC9 Q9UKV0 3/20 0.39
HDAC5 Q9UQL6 3/20 0.39
P2RY12 Q9H244 1/20 0.36
KDR P35968 3/20 0.36
S1PR2 O95136 1/20 0.36
SIRT5 Q9NXA8 1/20 0.36
MITF O75030 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7402346 0.89 HDAC1 (0.44) HDAC1HDAC4HDAC2HDAC8HDAC3
SCHEMBL7409694 0.86 MMP2 (0.42) HDAC1HDAC4HDAC2HDAC8HDAC3
SCHEMBL7410624 0.85 HDAC4 (0.41) HDAC1HDAC4HDAC2HDAC8HDAC3
SCHEMBL7406759 0.83 MMP2 (0.41) HDAC1HDAC4HDAC2HDAC8HDAC3
SCHEMBL7408851 0.83 MMP2 (0.41) HDAC1HDAC4HDAC2HDAC8HDAC3
SCHEMBL7406281 0.81 HDAC4 (0.39) HDAC1HDAC4HDAC2HDAC8HDAC3
SCHEMBL7409752 0.81 MMP3 (0.40) HDAC1HDAC4HDAC2HDAC8HDAC3
SCHEMBL7409945 0.78 F10 (0.41) HDAC1HDAC4HDAC2HDAC8HDAC3
SCHEMBL7407508 0.77 MMP3 (0.40) HDAC1HDAC4HDAC2HDAC8HDAC3
SCHEMBL7406513 0.76 MMP1 (0.42) HDAC1HDAC4HDAC2HDAC8HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed