SCHEMBL7405673

SCHEMBL7405673

COc1cc2c(C)nc(=O)n(CCC(=O)c3ccccc3)c2cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
HSD11B1 P28845 2/20 0.45
HTR1A P08908 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
MAPK1 P28482 1/20 0.41
THRB P10828 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2C P18825 1/20 0.41
MAPT P10636 4/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 2/20 0.40
GAA P10253 1/20 0.40
BLM P54132 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TSHR P16473 1/20 0.40
TP53 P04637 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL7404843 0.84 GPR35 (0.42) ALDH1A1HSD11B1KMT2AGAA
SCHEMBL7412075 0.82 DYRK1A (0.47) CTNNB1
SCHEMBL11128567 0.82 KDM4E (0.47) ALDH1A1HSD11B1MAPK1MEN1KMT2A
Water SCHEMBL10619090 0.81 KDM4E (0.46) ALDH1A1HSD11B1MAPK1MEN1KMT2A
SCHEMBL10985135 0.81 TNF (0.54) ALDH1A1
SCHEMBL7403886 0.80 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2MAPK1MAPTPOLB
SCHEMBL10974103 0.76 TNF (0.61) GAA
SCHEMBL7410167 0.76 MAPT (0.41) ALDH1A1SMN1; SMN2MAPK1THRBMAPT
SCHEMBL11076393 0.76 ACHE (0.48) ALDH1A1SMN1; SMN2MAPK1MAPTL3MBTL1
SCHEMBL10970598 0.76 TNF (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0107398-B1 ORTHO SUBSTITUTED DIHYDROXY-2(1H)QUINAZOLINONE-1-ALKANOIC ACIDS ORTHO PHARMA CORP (US) 1988-06-08 EP disclosed
US-4631283-A RENAL VASODILATORS, CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1986-12-23 US disclosed
US-4490374-A CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1984-12-25 US disclosed
EP-0107398-A1 Ortho substituted dihydroxy-2(1H)quinazolinone-1-alkanoic acids ORTHO PHARMACEUTICAL CORPORATION (US) 1984-05-02 EP disclosed