SCHEMBL7408564

SCHEMBL7408564

CC(C)CCN(C[C@@H](O)[C@H](Cc1ccccc1)NC(=O)CN(C(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1)C(C)(C)C)C(=O)NC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 1/20 0.44
KLK5 Q9Y337 1/20 0.41
PREP P48147 2/20 0.40
PRCP P42785 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
REN P00797 1/20 0.38
ACE P12821 2/20 0.38
GFER P55789 1/20 0.38
CTSD P07339 1/20 0.38
CTSE P14091 1/20 0.38
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7404180 0.92 KLK5 (0.46) KLK5ADORA3ADORA2AADORA2BADORA1
SCHEMBL7401649 0.82 CTRB1 (0.48) CTRB1PRCPTSHRL3MBTL1KDM4E
SCHEMBL7405664 0.81 BACE1 (0.38) KLK5RENCTSDCTSEBACE1
SCHEMBL7454378 0.81 BACE1 (0.38) KLK5RENCTSDCTSEBACE1
SCHEMBL7403106 0.80 PSEN1 (0.41) KLK5BACE1PSEN1PSEN2APH1B
SCHEMBL7399393 0.80 PSEN1 (0.41) KLK5BACE1PSEN1PSEN2APH1B
SCHEMBL7402855 0.79 PSEN1 (0.41) RENCTSDBACE1PSEN1PSEN2
SCHEMBL7400659 0.78 PSEN1 (0.42) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL6431948 0.78 CTSB (0.55) KLK5PSEN1PSEN2APH1BNCSTN
SCHEMBL6431945 0.78 CTSB (0.55) KLK5PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750648-A HUMAN IMMUNODEFICIENCY VIRUS G.D. SEARLE & CO. (US) 1998-05-12 US claimed
WO-1995006061-A1 RETROVIRAL PROTEASE INHIBITORS AND COMBINATIONS THEREOF G.D. SEARLE & CO. (US) 1995-03-02 WO claimed