SCHEMBL7409053

SCHEMBL7409053

Cc1ccc(OC[C@H]2CCN2)c(C(=O)N(C(N)=O)c2nc(C)ccc2OC[C@@H]2CCN2)n1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.39
CHRNB4 P30926 3/20 0.37
CHRNA3 P32297 3/20 0.37
CHRNB2 P17787 2/20 0.37
CHRNA5 P30532 1/20 0.37
CHRNA4 P43681 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415298 0.86 MAP2K1 (0.37) IRAK4CHRNB4CHRNA3
SCHEMBL7407282 0.83 CHRNA3 (0.44) IRAK4CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL7454988 0.81 CHRNA3 (0.39) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL7416819 0.79 MAP2K1 (0.45) IRAK4CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL7409579 0.79 CHRNB2 (0.44) IRAK4CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL7406760 0.76 CHRNB2 (0.45) CHRNB4CHRNA3CHRNB2CHRNA5CHRNA4
SCHEMBL7414935 0.74 CHRNA3 (0.39) IRAK4CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL7409488 0.72 CHRNB2 (0.55) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL7413684 0.69 CHRNB2 (0.48) CHRNB4CHRNA3CHRNB2CHRNA5CHRNA4
SCHEMBL7409563 0.69 CHRNB2 (0.48) CHRNB4CHRNA3CHRNB2CHRNA5CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047690-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-11-02 EP disclosed
WO-1999032480-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1999-07-01 WO disclosed