SCHEMBL7409495

SCHEMBL7409495

COc1cc(C=O)c(CCC(=O)O)c(C=O)c1O

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 13/20 0.46
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
P2RX3 P56373 2/20 0.41
PRKDC P78527 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417469 0.91 ERN1 (0.48) ERN1LMNAMAPTPRKDC
SCHEMBL15535074 0.82 ERN1 (0.49) ERN1LMNAMAPTPRKDCKDM4E
SCHEMBL16978281 0.81 ERN1 (0.51) ERN1LMNAMAPTPRKDCKDM4E
SCHEMBL7407211 0.81 P2RX3 (0.41) ERN1MAPTP2RX3KDM4EALDH1A1
SCHEMBL15547540 0.75 ERN1 (0.62) ERN1LMNAMAPTPRKDCKDM4E
SCHEMBL21933489 0.74 ERN1 (0.54) ERN1LMNAMAPTALDH1A1
SCHEMBL14925248 0.74 KDM4E (0.51) ERN1LMNAMAPTKDM4EALDH1A1
SCHEMBL7414964 0.74 MAPT (0.43) ERN1LMNAMAPTPRKDCKDM4E
SCHEMBL146097 0.73 ALDH1A1 (0.47) ALDH1A1TSHRTDP1
SCHEMBL9227782 0.72 TLR2 (0.53) ERN1LMNAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6150412-A SUCH AS 4-(5-HYDROXY-4-METHOXY-2-NITROPHENYL)BUTANOIC ACID; ADMINISTERING TO INHIBIT CATECHOL-O-METHYL TRANSFERASE; TREATING PARKINSON'S DISEASE OR HYPERTENSION ORION-YHTYMA OY (FI) 2000-11-21 US disclosed
WO-1996037456-A1 NEW CATECHOL DERIVATIVES Orion-Yhtymä Oy (FI) 1996-11-28 WO disclosed