SCHEMBL7414964

SCHEMBL7414964

COc1cc([N+](=O)[O-])c(CCCC(=O)O)c(C=O)c1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
PRKDC P78527 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ERN1 O75460 3/20 0.42
JUN P05412 1/20 0.40
IMPDH2 P12268 3/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
EGFR P00533 2/20 0.38
POLB P06746 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
GRK6 P43250 1/20 0.37
CTSD P07339 1/20 0.37
PTGDR Q13258 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7412241 0.84 IMPDH2 (0.41) MAPTJUNIMPDH2LMNAGAA
SCHEMBL7418340 0.84 XDH (0.42) MAPTKDM4EALDH1A1CYP3A4ALOX15
SCHEMBL7414973 0.81 IMPDH2 (0.40) MAPTALDH1A1JUNIMPDH2LMNA
SCHEMBL7408115 0.80 IMPDH2 (0.39) MAPTJUNIMPDH2LMNAGAA
SCHEMBL7417469 0.78 ERN1 (0.48) MAPTPRKDCERN1IMPDH2LMNA
SCHEMBL7410980 0.77 JUN (0.41) MAPTJUNIMPDH2HTTSMN1; SMN2
SCHEMBL7407867 0.75 CTSD (0.57) KDM4EALDH1A1CYP3A4LMNAHTT
SCHEMBL7414510 0.74 CTSD (0.49) KDM4EALDH1A1CYP3A4ALOX15IMPDH2
SCHEMBL7409495 0.74 ERN1 (0.46) MAPTKDM4EALDH1A1PRKDCERN1
SCHEMBL9252028 0.73 RAB9A (0.50) MAPTKDM4EALDH1A1JUNGRK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996033196-A1 INDOLE-3-CARBONYL AND INDOLE-3-SULFONYL DERIVATIVES AS PLATELET ACTIVATING FACTOR ANTAGONISTS ABBOTT LABORATORIES (US) 1996-10-24 WO claimed
US-6150412-A SUCH AS 4-(5-HYDROXY-4-METHOXY-2-NITROPHENYL)BUTANOIC ACID; ADMINISTERING TO INHIBIT CATECHOL-O-METHYL TRANSFERASE; TREATING PARKINSON'S DISEASE OR HYPERTENSION ORION-YHTYMA OY (FI) 2000-11-21 US disclosed
WO-1996037456-A1 NEW CATECHOL DERIVATIVES Orion-Yhtymä Oy (FI) 1996-11-28 WO disclosed