SCHEMBL7410095

SCHEMBL7410095

N=C(N)c1cccc(NC=O)c1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 12/20 0.49
PRSS2 P07478 5/20 0.49
PRSS3 P35030 5/20 0.49
F2 P00734 3/20 0.48
PLG P00747 2/20 0.48
C1S P09871 1/20 0.48
ALDH1A1 P00352 1/20 0.47
LOXL2 Q9Y4K0 1/20 0.46
PLAU P00749 1/20 0.44
PLAT P00750 1/20 0.44
KLKB1 P03952 1/20 0.44
KLK1 P06870 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8689035 0.85 PARP1 (0.55)
SCHEMBL171243 0.79 RAB9A (0.55) ALDH1A1
SCHEMBL7440442 0.79 PRSS1 (0.57) PRSS1PRSS2PRSS3F2ALDH1A1
SCHEMBL9335857 0.78 UNG (0.45) PRSS1PRSS2PRSS3F2PLG
SCHEMBL3901564 0.78 KMT2A (0.60) ALDH1A1
Amicarbalide SCHEMBL1818799 0.78 PLAU (0.65) PRSS1PRSS2PRSS3F2PLG
SCHEMBL11041250 0.78 ALDH1A1 (0.47) ALDH1A1
SCHEMBL12129057 0.77 ALDH1A1 (0.67) ALDH1A1
SCHEMBL10671451 0.77 PRSS1 (0.52) PRSS1PRSS2PRSS3F2PLG
SCHEMBL10177622 0.77 PRSS1 (0.52) PRSS1PRSS2PRSS3F2PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0542708-B1 Substituted beta-amino acid derivatives useful as platelet aggregation inhibitors MONSANTO CO (US) 2001-05-30 EP disclosed
WO-1993007867-A1 SUBSTITUTED β-AMINO ACID DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-04-29 WO disclosed