SCHEMBL7410339

SCHEMBL7410339

CN(C)C(=O)COP(=O)(CN[C@@H](Cc1ccc(-c2ccccc2)cc1)C(=O)O)OCC(=O)N(C)C

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MME P08473 12/20 0.45
ACE P12821 10/20 0.44
ACE2 Q9BYF1 9/20 0.44
CPA1 P15085 7/20 0.44
GPR34 Q9UPC5 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7413312 0.85 MME (0.45) MMEACEACE2CPA1GPR34
SCHEMBL7408519 0.83 MAPT (0.49) MMEACEACE2CPA1GPR34
SCHEMBL7322712 0.82 MME (0.51) MMEACEACE2CPA1
SCHEMBL7348038 0.82 MME (0.51) MMEACEACE2CPA1
SCHEMBL3103119 0.80 FPR2 (0.54) MMEACEACE2CPA1
SCHEMBL8922274 0.80 MME (0.47) MME
SCHEMBL8922261 0.80 MME (0.47) MME
SCHEMBL7414929 0.79 MME (0.45) MMEACEACE2CPA1GPR34
SCHEMBL7407175 0.78 MME (0.48) MMEACEACE2CPA1
SCHEMBL7411127 0.76 MME (0.62) MMEACEACE2CPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660840-B1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA GEIGY AG (CH) 1997-05-07 EP disclosed
US-5550119-A ENDOTHELIN-CONVERTING ENZYM INHIBITORS CIBA-GEIGY CORPORATION (US) 1996-08-27 US disclosed
EP-0660840-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES. CIBA GEIGY AG (CH) 1995-07-05 EP disclosed
WO-1994005677-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1994-03-17 WO disclosed
US-5250522-A Neutral endopeptidase inhibitors; cardiovascular disorders CIBA-GEIGY CORPORATION (US) 1993-10-05 US disclosed