SCHEMBL7407175

SCHEMBL7407175

O=C(O)[C@H](Cc1ccc(-c2ccccc2)cc1)NCP(=O)(Oc1ccccc1)Oc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MME P08473 9/20 0.48
PPARG P37231 6/20 0.48
PPARA Q07869 5/20 0.48
ACE2 Q9BYF1 7/20 0.47
ACE P12821 7/20 0.47
CPA1 P15085 5/20 0.47
SRR Q9GZT4 1/20 0.46
PSAT1 Q9Y617 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31510352 0.93 ANPEP (0.48) MMEACE2ACECPA1
SCHEMBL7419794 0.90 MME (0.50) MME
SCHEMBL7415659 0.89 KMT2A (0.48) MMEACE2ACECPA1
SCHEMBL7413775 0.89 PPARG (0.49) MMEPPARGPPARAACE2ACE
SCHEMBL8932450 0.88 MME (0.47) MMEPPARGPPARAACE2ACE
SCHEMBL7412181 0.88 MME (0.44) MMEPPARGPPARAACE2ACE
SCHEMBL7466186 0.88 FPR2 (0.47) MMEPPARGPPARAACE2ACE
SCHEMBL7415833 0.87 ITGA4 (0.55) PPARGPPARA
SCHEMBL7404577 0.87 F2 (0.47) PPARGPPARAACE
SCHEMBL7310756 0.86 MME (0.55) MMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660840-B1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA GEIGY AG (CH) 1997-05-07 EP claimed
EP-0660840-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES. CIBA GEIGY AG (CH) 1995-07-05 EP claimed
WO-1994005677-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1994-03-17 WO claimed
US-5250522-A Neutral endopeptidase inhibitors; cardiovascular disorders CIBA-GEIGY CORPORATION (US) 1993-10-05 US claimed
EP-0660840-B1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA GEIGY AG (CH) 1997-05-07 EP disclosed
WO-1996026729-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES AS ECE INHIBITORS CIBA-GEIGY AG (CH) 1996-09-06 WO disclosed
US-5550119-A ENDOTHELIN-CONVERTING ENZYM INHIBITORS CIBA-GEIGY CORPORATION (US) 1996-08-27 US disclosed
EP-0660840-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES. CIBA GEIGY AG (CH) 1995-07-05 EP disclosed
WO-1994005677-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1994-03-17 WO disclosed
US-5250522-A Neutral endopeptidase inhibitors; cardiovascular disorders CIBA-GEIGY CORPORATION (US) 1993-10-05 US disclosed