SCHEMBL7410402

SCHEMBL7410402

COc1cccc2[nH]c3c(c12)CC(N(C)C)CC3

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 2/20 0.59
CHRM2 P08172 1/20 0.59
CHRM1 P11229 1/20 0.59
DRD2 P14416 2/20 0.54
DRD4 P21917 1/20 0.54
DRD3 P35462 1/20 0.54
HTR2C P28335 2/20 0.50
HTR1A P08908 1/20 0.49
ADRA1A P35348 1/20 0.44
MAPKAPK2 P49137 1/20 0.43
MAPK10 P53779 1/20 0.42
RIPK1 Q13546 1/20 0.42
HTR1F P30939 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410925 0.83 CHRM3 (0.43) CHRM3CHRM2CHRM1DRD2DRD4
SCHEMBL7460577 0.83 HTR2A (0.43) CHRM3CHRM2CHRM1DRD2DRD4
Hydrochloric Acid SCHEMBL7407711 0.82 HTR2A (0.43) CHRM3CHRM2CHRM1DRD2DRD4
SCHEMBL24408232 0.82 NR2E1 (0.56) DRD2DRD3HTR2CADRA1AMAPKAPK2
SCHEMBL7405543 0.82 HTR1A (0.47) CHRM3CHRM2CHRM1DRD2DRD4
SCHEMBL7408361 0.82 HTR1A (0.50) CHRM3CHRM2CHRM1HTR1AHTR1F
Hydrochloric Acid SCHEMBL7410552 0.81 CHRM3 (0.55) CHRM3CHRM2CHRM1DRD2DRD4
SCHEMBL7412749 0.80 HTR1F (0.41) CHRM3CHRM2CHRM1DRD2DRD4
SCHEMBL7408846 0.80 HTR1F (0.41) CHRM3CHRM2CHRM1DRD2DRD4
SCHEMBL4904443 0.80 HTR2C (0.47) CHRM3CHRM2CHRM1HTR2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4257952-A PSYCHOTROPIC DRUGS, ANALGESICS, ANTIHISTAMINES STERLING DRUG INC. (US) 1981-03-24 US disclosed
US-4172834-A ANALGESICS, ANTIHISTAMINES AND PSYCHOTROPIC AGENTS STERLING DRUG INC. (US) 1979-10-30 US disclosed
US-4062864-A ANALGESIC, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1977-12-13 US disclosed
US-3959309-A ANALGESICS, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1976-05-25 US disclosed