SCHEMBL7410707

SCHEMBL7410707

COc1ccc(C(=O)NC(C(=O)O)C(C)C)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.71
PPARG P37231 2/20 0.63
PPARA Q07869 1/20 0.63
DGAT1 O75907 1/20 0.62
CA2 P00918 4/20 0.60
CA1 P00915 3/20 0.60
MMP2 P08253 2/20 0.57
MMP9 P14780 2/20 0.57
ALDH1A1 P00352 2/20 0.56
TAS1R3 Q7RTX0 1/20 0.55
TAS1R1 Q7RTX1 1/20 0.55
PLK1 P53350 1/20 0.54
LMNA P02545 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
MMP1 P03956 1/20 0.52
MMP3 P08254 1/20 0.52
MMP7 P09237 1/20 0.52
MMP8 P22894 1/20 0.52
MMP13 P45452 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5838728 1.00 NPSR1 (0.71) NPSR1PPARGPPARADGAT1CA2
SCHEMBL11509188 0.95 NPSR1 (0.66) NPSR1PPARGPPARADGAT1CA2
SCHEMBL9828979 0.89 NPSR1 (0.57) NPSR1PPARGPPARADGAT1CA2
SCHEMBL9828975 0.89 NPSR1 (0.57) NPSR1PPARGPPARADGAT1CA2
SCHEMBL10659164 0.88 NPSR1 (0.56) NPSR1PPARGPPARADGAT1CA2
SCHEMBL10659171 0.88 NPSR1 (0.56) NPSR1PPARGPPARADGAT1CA2
SCHEMBL15906297 0.87 ALDH1A1 (0.60) NPSR1DGAT1CA2CA1ALDH1A1
SCHEMBL21274384 0.85 CA2 (0.64) NPSR1PPARGPPARADGAT1CA2
SCHEMBL21274381 0.85 CA2 (0.64) NPSR1PPARGPPARADGAT1CA2
SCHEMBL11509003 0.84 NPSR1 (0.68) NPSR1PPARGPPARADGAT1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112261939-A Granzyme B directed imaging and therapy 塞托赛特生物制药股份有限公司 2021-01-22 CN disclosed
WO-2018011230-A1 PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR GAMMA AGONISTS, METHOD OF PREPARATION AND USES THEREOF UNIVERSITE D'AIX-MARSEILLE (FR) 2018-01-18 WO disclosed
EP-1140846-A1 ASPARTIC PROTEASE INHIBITORS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2001-10-10 EP disclosed
WO-2000040558-A1 ASPARTIC PROTEASE INHIBITORS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-07-13 WO disclosed