SCHEMBL7410732

SCHEMBL7410732

CC(C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](C)NC(=O)[C@H](C)N1C(=O)CCC1=O)C(=O)N([N+]=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ELANE P08246 17/20 0.43
XIAP P98170 1/20 0.40
MLX Q9UH92 1/20 0.40
CMA1 P23946 1/20 0.39
ACE P12821 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540221 0.88 TACR1 (0.48) CMA1ACE
SCHEMBL8662695 0.87 ELANE (0.45) ELANEXIAPMLXCMA1
SCHEMBL7400531 0.83 ELANE (0.47) ELANEXIAPMLX
SCHEMBL7874280 0.83 EPHA2 (0.43) ACE
SCHEMBL6057548 0.82 XIAP (0.46) ELANEXIAPMLXCMA1ACE
SCHEMBL5494650 0.82 ELANE (0.40) ELANEXIAPMLXCMA1
SCHEMBL10895690 0.81 ELANE (0.42) ELANECMA1
SCHEMBL8333459 0.80 PSMB9 (0.47) XIAP
SCHEMBL1289940 0.79 CMA1 (0.54) ELANEXIAPCMA1ACE
SCHEMBL8660922 0.77 ELANE (0.39) ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189901-A1 OXAZAHETEROCYCLES AS PROTEASE INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2002-03-27 EP disclosed
WO-2000073302-A1 OXAZAHETEROCYCLES AS PROTEASE INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-12-07 WO disclosed