SCHEMBL741162

SCHEMBL741162

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc(Br)cc3)NC(=O)O)C2)nc2c(Cl)cccc21

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 1/20 0.35
ALDH1A1 P00352 2/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
HRH1 P35367 3/20 0.34
CYP2D6 P10635 2/20 0.34
ITK Q08881 1/20 0.34
KCNH2 Q12809 3/20 0.34
REN P00797 4/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
ALOX5AP P20292 2/20 0.33
HSD11B1 P28845 2/20 0.33
ITGB1 P05556 2/20 0.33
ITGA5 P08648 1/20 0.33
CHRM1 P11229 1/20 0.33
ITGA4 P13612 1/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741369 0.93 MMEL1 (0.38) ALDH1A1TSHRKMT2AHRH1CYP2D6
SCHEMBL763266 0.91 KLK5 (0.35) ALDH1A1TSHRKMT2AHRH1CYP2D6
SCHEMBL739361 0.89 HRH1 (0.35) FPR2ALDH1A1TSHRKMT2AHRH1
SCHEMBL739919 0.89 HRH1 (0.45) HRH1CYP2D6KCNH2CHRM1
SCHEMBL762867 0.85 HRH2 (0.37) KMT2AHRH1ITGB3ITGA2B
SCHEMBL740312 0.84 HRH1 (0.45) HRH1CYP2D6KCNH2CHRM1
SCHEMBL742017 0.84 NLRP3 (0.41) ALDH1A1TSHRKMT2AHRH1CYP2D6
SCHEMBL740291 0.83 DPP4 (0.37) ALDH1A1TSHRKMT2AHRH1CYP2D6
SCHEMBL740290 0.83 DPP4 (0.37) ALDH1A1TSHRKMT2AHRH1CYP2D6
SCHEMBL2791612 0.83 PROKR1 (0.39) FPR2ALDH1A1TSHRKMT2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed