SCHEMBL7412459

SCHEMBL7412459

CCOC(=O)C[C@@H](NC1CCC1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.41
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP2D6 P10635 1/20 0.40
GAA P10253 2/20 0.38
MGAM O43451 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
CASP6 P55212 1/20 0.36
TP53 P04637 2/20 0.35
LMNA P02545 2/20 0.35
SMYD3 Q9H7B4 1/20 0.35
TSHR P16473 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KMT2A Q03164 1/20 0.34
HTT P42858 1/20 0.34
UGT2B7 P16662 2/20 0.34
PPM1B O75688 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7377849 1.00 THRB (0.41) THRBATML3MBTL1CYP2D6GAA
SCHEMBL7379026 0.97 THRB (0.44) THRBATML3MBTL1CYP2D6GAA
SCHEMBL7380230 0.85 EPHX2 (0.39) CYP2D6LMNAALDH1A1
SCHEMBL7525610 0.81 LMNA (0.35) CYP2D6LMNATSHRALDH1A1MAPT
SCHEMBL12482729 0.78 LMNA (0.41) THRBATML3MBTL1KDM4ELMNA
SCHEMBL3668494 0.78 CYP2D6 (0.48) THRBATML3MBTL1CYP2D6GAA
SCHEMBL20614287 0.77 CYP2D6 (0.38) THRBATML3MBTL1CYP2D6GAA
SCHEMBL38057 0.77 EPHX1 (0.40) CYP2D6GAALMNA
SCHEMBL38058 0.77 EPHX1 (0.40) CYP2D6GAALMNA
SCHEMBL16439931 0.76 LMNA (0.40) THRBATML3MBTL1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922054-B1 ANTICOAGULANT PEPTIDYL-ARGININE ALDEHYDE DERIVATIVES GYOGYSZERKUTATO INTEZET (HU) 2002-08-14 EP disclosed
US-6235707-B1 Anticoagulant peptidyl-arginine aldehyde derivatives GYOGYSZERKUTATO INTEZET KFT. (HU) 2001-05-22 US disclosed
EP-0922054-A1 ANTICOAGULANT PEPTIDYL-ARGININE ALDEHYDE DERIVATIVES GYOGYSZERKUTATO INTEZET KFT. (HU) 1999-06-16 EP disclosed
WO-1997046576-A1 ANTICOAGULANT PEPTIDYL-ARGININE ALDEHYDE DERIVATIVES Gyógyszerkutató Intézet Kft. (HU) 1997-12-11 WO disclosed