SCHEMBL7412588

SCHEMBL7412588

O=C1CCC(OC(=O)c2cccc(C(F)(F)F)c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56
HPGD P15428 2/20 0.56
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 1/20 0.56
CES2 O00748 2/20 0.50
KMT2A Q03164 2/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
LMNA P02545 3/20 0.44
POLB P06746 1/20 0.44
HSD11B1 P28845 1/20 0.44
SRD5A2 P31213 1/20 0.43
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
TAS1R2 Q8TE23 1/20 0.43
MEN1 O00255 1/20 0.42
P2RX1 P51575 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9299353 0.87 HPGD (0.60) CYP2C9CYP2C19HPGDKDM4EALDH1A1
SCHEMBL28968096 0.84 ALDH1A1 (0.56) CYP2C9CYP2C19HPGDKDM4EALDH1A1
SCHEMBL18455052 0.82 CYP2C9 (0.54) CYP2C9CYP2C19HPGDKDM4EALDH1A1
SCHEMBL28342942 0.79 HPGD (0.52) CYP2C9CYP2C19HPGDKDM4EALDH1A1
SCHEMBL1556598 0.78 MEN1 (0.59) CYP2C9CYP2C19KMT2AGAAMAPT
SCHEMBL28637086 0.76 CES2 (0.54) CYP2C9CYP2C19HPGDKDM4EALDH1A1
SCHEMBL11802784 0.76 CES2 (0.67) HPGDKDM4EALDH1A1CES2KMT2A
SCHEMBL11047986 0.75 CYP2C9 (0.48) CYP2C9CYP2C19HPGDKDM4EALDH1A1
SCHEMBL8633064 0.74 SLC6A2 (0.59) KDM4EKMT2AMEN1
SCHEMBL31406174 0.74 CES2 (0.69) HPGDALDH1A1CES2KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4257952-A PSYCHOTROPIC DRUGS, ANALGESICS, ANTIHISTAMINES STERLING DRUG INC. (US) 1981-03-24 US disclosed
US-4172834-A ANALGESICS, ANTIHISTAMINES AND PSYCHOTROPIC AGENTS STERLING DRUG INC. (US) 1979-10-30 US disclosed
US-4062864-A ANALGESIC, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1977-12-13 US disclosed
US-3959309-A ANALGESICS, PSYCHOTROPIC, ANTIHISTAMINE STERLING DRUG INC. (US) 1976-05-25 US disclosed