SCHEMBL7412781

SCHEMBL7412781

Cc1ccc(C)c(S(=O)(=O)N[C@@H](Cc2ccc(OCCCONC(=N)N)cc2)C(=O)O)c1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.53
ITGB3 P05106 13/20 0.52
ITGA2B P08514 11/20 0.52
ALDH1A1 P00352 1/20 0.51
CYP2C19 P33261 1/20 0.51
ITGB1 P05556 1/20 0.44
ITGA4 P13612 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
POLB P06746 1/20 0.43
PPARG P37231 1/20 0.42
ITGAV P06756 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7410411 0.96 L3MBTL1 (0.49) L3MBTL1ITGB3ITGA2BALDH1A1CYP2C19
SCHEMBL7413005 0.91 ITGB3 (0.50) L3MBTL1ITGB3ITGA2BALDH1A1CYP2C19
SCHEMBL7695352 0.90 ITGB3 (0.49) L3MBTL1ITGB3ITGA2BCYP2C19ITGB1
Trifluoroacetic Acid SCHEMBL7413938 0.88 ITGB3 (0.47) L3MBTL1ITGB3ITGA2BCYP2C19ITGB1
SCHEMBL7409539 0.88 ITGB3 (0.47) L3MBTL1ITGB3ITGA2BITGB1ITGA4
SCHEMBL7410553 0.88 ITGB3 (0.50) ITGB3ITGA2BITGB1ITGA4POLB
SCHEMBL7418575 0.87 ITGB3 (0.55) ITGB3ITGA2BITGB1ITGA4ITGAV
SCHEMBL7411712 0.87 TDP1 (0.59) L3MBTL1ITGB3ITGA2BTDP1
SCHEMBL7410416 0.87 L3MBTL1 (0.41) L3MBTL1ITGB3ITGA2BALDH1A1CYP2C19
Trifluoroacetic Acid SCHEMBL7419764 0.87 CYP3A4 (0.47) L3MBTL1ITGB3ITGA2BCYP2C19ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US claimed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP claimed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO claimed