SCHEMBL7412860

SCHEMBL7412860

Cc1nn(C)c(C)c1C[CH]CC(N)=O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 4/20 0.38
GAA P10253 2/20 0.38
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
LMNA P02545 1/20 0.36
TTR P02766 1/20 0.34
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7374141 0.76 KDM4E (0.47) KDM4EALDH1A1GAARAB9ANPC1
SCHEMBL1778339 0.73 SMN1; SMN2 (0.44) KDM4EALDH1A1GAARAB9ANPC1
SCHEMBL11562262 0.72 KDM4E (0.44) KDM4EALDH1A1GAARAB9ANPC1
SCHEMBL4891782 0.69 KDM4E (0.43) KDM4EALDH1A1GAARAB9ANPC1
SCHEMBL7417039 0.69 KMT2A (0.38) ALDH1A1GAAKMT2A
SCHEMBL4353356 0.68 ALDH1A1 (0.46) KDM4EALDH1A1GAARAB9ANPC1
SCHEMBL7382372 0.68 RAF1 (0.34)
SCHEMBL7379327 0.67 MPO (0.34)
SCHEMBL762264 0.67 SMN1; SMN2 (0.43) KDM4EALDH1A1GAARAB9ANPC1
SCHEMBL5898267 0.67 SMN1; SMN2 (0.47) KDM4EALDH1A1GAARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165500-A1 AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES,TNF-ALPHA,AND AGGRECANASE Du Pont Pharmaceuticals Company (US) 2002-01-02 EP disclosed
WO-2000059874-A1 NOVEL AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES, TNF-α, AND AGGRECANASE DU PONT PHARMACEUTICALS COMPANY (US) 2000-10-12 WO disclosed