SCHEMBL7412892

SCHEMBL7412892

COC(=O)C(CCC(=O)OC(C)(C)C)NC(=O)C(CC(C)C)C(=O)NC(C=O)CC(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MME P08473 1/20 0.39
CTSB P07858 2/20 0.37
BIRC2 Q13490 3/20 0.36
MMP1 P03956 1/20 0.35
CTSK P43235 4/20 0.34
CTSL P07711 2/20 0.32
CTSS P25774 1/20 0.32
CYP2D6 P10635 1/20 0.32
FOLH1 Q04609 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7404509 0.90 MME (0.40) MMECTSBMMP1CTSKCTSL
SCHEMBL7448782 0.82 CTSB (0.42) CTSB
SCHEMBL7406391 0.81 CTSB (0.44) MMECTSBMMP1CTSKCTSL
SCHEMBL7409805 0.80 CTSB (0.46) MMECTSBCTSKCTSLCTSS
SCHEMBL7406513 0.80 MMP1 (0.42) MMP1CTSK
SCHEMBL7406281 0.75 HDAC4 (0.39) CTSBMMP1CTSK
SCHEMBL5489915 0.74 CTSK (0.39) CTSBMMP1CTSKCTSLCTSS
SCHEMBL16024776 0.73 PSMB5 (0.40) CTSBCTSKCTSLCTSS
SCHEMBL8254105 0.72 FOLH1 (0.40) CTSBBIRC2CTSKCTSLCTSS
SCHEMBL18161574 0.71 CYP2D6 (0.40) CTSBMMP1CTSKCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed