SCHEMBL7413495

SCHEMBL7413495

Cc1cccc2[nH]c(C3CCN(C4CCN(C)CC4)CC3)nc12

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 0.58
PARP2 Q9UGN5 3/20 0.50
HRH4 Q9H3N8 1/20 0.46
PDE10A Q9Y233 1/20 0.43
PKM P14618 1/20 0.42
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
TLR9 Q9NR96 1/20 0.41
TLR7 Q9NYK1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5621269 0.82 PARP1 (0.87) PARP1PARP2
SCHEMBL4374769 0.81 ALDH1A1 (0.53) PARP1PARP2PDE10A
Hydrochloric Acid SCHEMBL18614325 0.81 PARP1 (0.85) PARP1PARP2
SCHEMBL6869690 0.80 PARP1 (0.62) PARP1PARP2
SCHEMBL7409877 0.77 PARP1 (0.55) PARP1PARP2HRH4
SCHEMBL7469714 0.76 PARP1 (0.53) PARP1PARP2PDE10APTGS1PTGS2
SCHEMBL7215446 0.76 PARP1 (0.61) PARP1PARP2PDE10A
SCHEMBL6646211 0.75 PARP14 (0.61) PARP1PARP2
SCHEMBL5621887 0.73 PARP1 (1.00) PARP1PARP2
SCHEMBL19127880 0.72 PARP1 (0.53) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed