SCHEMBL7469714

SCHEMBL7469714

Cc1cccc2[nH]c(C3CCN(CCC(C)C)CC3)nc12

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.53
PARP2 Q9UGN5 2/20 0.53
PDE10A Q9Y233 1/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
NPY1R P25929 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5621431 0.83 PARP1 (0.79) PARP1PARP2
Hydrochloric Acid SCHEMBL7702646 0.82 PARP1 (0.78) PARP1PARP2
SCHEMBL6874947 0.80 PARP1 (0.58) PARP1PARP2
SCHEMBL4374769 0.79 ALDH1A1 (0.53) PARP1PARP2PDE10A
SCHEMBL7413495 0.76 PARP1 (0.58) PARP1PARP2PDE10APTGS1PTGS2
SCHEMBL7215446 0.74 PARP1 (0.61) PARP1PARP2PDE10A
SCHEMBL20463361 0.74 PARP1 (0.46) PARP1PARP2PDE10APTGS1PTGS2
SCHEMBL7460929 0.72 PARP1 (0.55) PARP1PTGS1PTGS2
SCHEMBL5620099 0.71 PARP1 (0.76) PARP1PARP2
SCHEMBL7524606 0.71 ALDH1A1 (0.45) PARP1PARP2PDE10APTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed