SCHEMBL7413588

SCHEMBL7413588

O=P(O)(O)C(NS(=O)(=O)c1ccc(-c2ccc(Cl)cc2)cc1)c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 13/20 0.66
CA12 O43570 6/20 0.66
CA9 Q16790 6/20 0.66
CA14 Q9ULX7 6/20 0.66
CA2 P00918 5/20 0.66
MMP8 P22894 4/20 0.66
CA1 P00915 4/20 0.66
MMP9 P14780 5/20 0.60
MMP1 P03956 4/20 0.60
MMP3 P08254 4/20 0.60
MMP7 P09237 4/20 0.60
MMP13 P45452 4/20 0.60
MMP14 P50281 3/20 0.60
ADAMTS5 Q9UNA0 1/20 0.53
FLT1 P17948 2/20 0.47
FLT4 P35916 2/20 0.47
KDR P35968 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
ADAMTS4 O75173 1/20 0.46
CYP1A2 P05177 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7413590 1.00 MMP2 (0.66) MMP2CA12CA9CA14CA2
SCHEMBL7656970 0.83 MMP2 (0.52) MMP2CA12CA9CA14CA2
SCHEMBL7968315 0.83 CASP1 (0.45) MMP2CA12CA9CA14CA2
SCHEMBL7968317 0.83 CASP1 (0.45) MMP2CA12CA9CA14CA2
SCHEMBL7409478 0.77 MMP2 (0.74) MMP2CA12CA9CA14CA2
SCHEMBL7409476 0.77 MMP2 (0.74) MMP2CA12CA9CA14CA2
SCHEMBL7648573 0.75 MMP2 (1.00) MMP2CA12CA9CA14CA2
SCHEMBL7648565 0.75 MMP2 (1.00) MMP2CA12CA9CA14CA2
SCHEMBL14602254 0.75 MMP2 (0.67) MMP2MMP9MMP1MMP3MMP7
SCHEMBL9435889 0.75 MMP2 (1.00) MMP2CA12CA9CA14CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1097159-B1 PHOSPHINOUS AND PHOSPHONIC ACID DERIVATIVES USED AS MEDICAMENTS AVENTIS PHARMA GMBH (DE) 2002-11-06 EP claimed
US-6500811-B2 PROPHYLAXIS AND THERAPY OF DISORDERS IN THE COURSE OF WHICH AN INCREASED ACTIVITY OF MATRIX-DEGRADING ENZYMES IS INVOLVED; THESE INCLUDE DEGENERATIVE JOINT DISORDERS SUCH AS OSTEOARTHROSES AND DISORDERS OF CONNECTIVE TISSUE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-12-31 US disclosed
EP-1097159-B1 PHOSPHINOUS AND PHOSPHONIC ACID DERIVATIVES USED AS MEDICAMENTS AVENTIS PHARMA GMBH (DE) 2002-11-06 EP disclosed
US-20020082246-A1 Sulfonylaminophosphinic and sulfonylaminophosphonic acid derivatives, methods for their preparation and use AVENTIS PHARMA DEUTSCHLAND GMBH. 2002-06-27 US disclosed
US-6235727-B1 ENZYME INHIBITORS; MUSCULAR DISORDERS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-05-22 US disclosed
EP-1097159-A1 PHOSPHINOUS AND PHOSPHONIC ACID DERIVATIVES USED AS MEDICAMENTS Aventis Pharma Deutschland GmbH (DE) 2001-05-09 EP disclosed
WO-2000004030-A1 PHOSPHINOUS AND PHOSPHONIC ACID DERIVATIVES USED AS MEDICAMENTS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-01-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020082246-A1 Sulfonylaminophosphinic and sulfonylaminophosphonic acid derivatives, methods for their preparation and use ARSA, STS, PNPO MMP2 24/4885CA12 1117/4885CA9 533/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.