SCHEMBL7414221

SCHEMBL7414221

N[C@@H](Cc1ccc(C(=O)C2CNCCO2)cc1)C(=O)N[C@@H](CCc1ccccc1)S(=O)(=O)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CTSC P53634 7/20 0.37
CTSB P07858 2/20 0.37
CTSH P09668 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
SSTR4 P31391 1/20 0.35
CTSL P07711 1/20 0.34
GHSR Q92847 1/20 0.34
MMP2 P08253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696045 1.00 CA2 (0.38) CA2CA12CA1CTSCCTSB
SCHEMBL8159878 0.90 CTSC (0.36) CA2CA12CA1CTSCCTSB
SCHEMBL7355598 0.86 CTSB (0.56) CTSCCTSBCTSHCTSSCTSK
SCHEMBL7349455 0.86 CTSB (0.56) CTSCCTSBCTSHCTSSCTSK
SCHEMBL7411057 0.83 CTSC (0.37) CTSCSSTR4GHSR
Hydrochloric Acid SCHEMBL7405421 0.83 CTSC (0.37) CTSCCTSBCTSHCTSSCTSK
SCHEMBL7414186 0.83 CTSC (0.33) CA2CA12CA1CTSCCTSB
SCHEMBL7352317 0.83 CTSB (0.48) CTSCCTSBCTSHCTSSCTSK
SCHEMBL7350474 0.82 CTSL (0.44) CTSCCTSBCTSHCTSSCTSK
SCHEMBL7410507 0.81 CTSC (0.36) CTSCSSTR4GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776718-A Reversible protease inhibitors ARRIS PHARMACEUTICAL CORPORATION (US) 1998-07-07 US disclosed
EP-0817778-A1 REVERSIBLE PROTEASE INHIBITORS ARRIS PHARMACEUTICAL CORPORATION (US) 1998-01-14 EP disclosed
WO-1996030353-A1 REVERSIBLE PROTEASE INHIBITORS ARRIS PHARMACEUTICAL CORPORATION (US) 1996-10-03 WO disclosed