SCHEMBL7414875

SCHEMBL7414875

O=C1NCc2cc(Br)ncc2N1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.46
CYP11B2 P19099 2/20 0.46
MB P02144 1/20 0.45
PDE3B Q13370 2/20 0.44
PDE3A Q14432 2/20 0.44
MAPK1 P28482 1/20 0.42
CRBN Q96SW2 1/20 0.34
CMA1 P23946 1/20 0.32
AHR P35869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25300707 0.75 AHR (0.49) CYP11B1CYP11B2PDE3BPDE3ACRBN
SCHEMBL429197 0.71 PDE3B (0.58) CYP11B1CYP11B2MBPDE3BPDE3A
SCHEMBL25242815 0.71 MKNK2 (0.45)
SCHEMBL24680963 0.71 CYP11B1 (0.46) CYP11B1CYP11B2PDE3BPDE3A
SCHEMBL16318310 0.69 CMA1 (0.59) CYP11B1CYP11B2MBPDE3BPDE3A
SCHEMBL6684530 0.69 CYP11B1 (0.53) CYP11B1CYP11B2MBPDE3BPDE3A
SCHEMBL31173261 0.69 CMA1 (0.59) CYP11B1CYP11B2MBPDE3BPDE3A
SCHEMBL23302034 0.69 MB (0.49) CYP11B1CYP11B2MBPDE3BPDE3A
SCHEMBL7419264 0.69 BIRC2 (0.37) CYP11B1CYP11B2MBPDE3BPDE3A
SCHEMBL15951381 0.69 MB (0.66) CYP11B1CYP11B2MBPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0333727-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (a Delaware corporation) (US) 1989-09-27 EP disclosed
US-4859672-A Pyrido[2,3-d]pyrimidinone and imidazo[4,5-b]pyrimidinone RORER PHARMACEUTICAL CORPORATION (US) 1989-08-22 US disclosed
WO-1988003025-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (US) 1988-05-05 WO disclosed