SCHEMBL7419264

SCHEMBL7419264

O=C1NCc2nc(Br)ncc2N1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BIRC2 Q13490 1/20 0.37
MB P02144 1/20 0.35
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
PARP16 Q8N5Y8 1/20 0.31
PARP3 Q9Y6F1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL674111 0.71 CYP11B1 (0.38) BIRC2MBCYP11B1CYP11B2PDE3B
SCHEMBL7414875 0.69 CYP11B1 (0.46) MBCYP11B1CYP11B2PDE3BPDE3A
SCHEMBL7420481 0.69 MB (0.45) MBPARP16PARP3
SCHEMBL673377 0.66 CYP11B1 (0.42) BIRC2MBCYP11B1CYP11B2PDE3B
SCHEMBL21146603 0.63 PDE3B (0.38) BIRC2MBCYP11B1CYP11B2PDE3B
SCHEMBL336931 0.62 MB (0.44) BIRC2MB
SCHEMBL23272058 0.62 BIRC2 (0.40) BIRC2MBCYP11B1CYP11B2PDE3B
SCHEMBL22686202 0.61 BIRC2 (0.39) BIRC2MBCYP11B1CYP11B2PDE3B
SCHEMBL2183634 0.61 POLB (0.51)
SCHEMBL11078154 0.59 MB (0.35) MB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5002944-A Compounds having cardiotonic activity RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-03-26 US disclosed
EP-0333727-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (a Delaware corporation) (US) 1989-09-27 EP disclosed
US-4859672-A Pyrido[2,3-d]pyrimidinone and imidazo[4,5-b]pyrimidinone RORER PHARMACEUTICAL CORPORATION (US) 1989-08-22 US disclosed
WO-1988003025-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (US) 1988-05-05 WO disclosed