SCHEMBL7415329

SCHEMBL7415329

Cc1cc(Cl)cc(Cl)c1S(=O)(=O)N[C@@H](Cc1ccc(OCCCONC(=N)N)cc1)C(=O)OC(=O)C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.35
ITGA2B P08514 6/20 0.35
ITGAV P06756 5/20 0.35
AVPR1A P37288 6/20 0.34
ITGB1 P05556 1/20 0.34
ITGA5 P08648 1/20 0.34
NR3C1 P04150 1/20 0.33
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415220 0.95 ITGB1 (0.36) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7422540 0.91 ITGB3 (0.42) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7408422 0.90 ITGB1 (0.40) ITGB3ITGA2BITGAVITGB1ITGA5
Trifluoroacetic Acid SCHEMBL7415325 0.90 ITGB3 (0.44) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7415327 0.88 ITGB1 (0.42) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7416602 0.88 ITGB3 (0.38) ITGB3ITGA2BITGAVITGB1ITGA5
SCHEMBL7417563 0.88 ITGB3 (0.39) ITGB3ITGA2BITGAV
SCHEMBL7408394 0.88 ITGB3 (0.37) ITGB3ITGA2BITGB1ITGA5PPARA
SCHEMBL7412118 0.88 ACLY (0.38) ITGB3ITGA2BITGB1ITGA5PPARA
SCHEMBL7416087 0.88 POLB (0.37) ITGB3ITGA2BITGAVITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed