SCHEMBL7416602

SCHEMBL7416602

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2cc(Cl)cc(Cl)c2)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.38
ITGA2B P08514 11/20 0.38
F2 P00734 7/20 0.38
TMPRSS6 Q8IU80 7/20 0.38
ITGAV P06756 5/20 0.36
ITGB1 P05556 1/20 0.35
ITGA5 P08648 1/20 0.35
RHOC P08134 1/20 0.33
RHOA P61586 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415008 0.93 F2 (0.42) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7414434 0.92 F2 (0.42) ITGB3ITGA2BF2TMPRSS6RHOC
SCHEMBL7415220 0.91 ITGB1 (0.36) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7415413 0.90 TMPRSS6 (0.38) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7412728 0.89 F2 (0.39) ITGB3ITGA2BF2TMPRSS6ITGAV
Trifluoroacetic Acid SCHEMBL7416599 0.89 ITGB3 (0.47) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7417592 0.89 ITGB3 (0.49) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7415235 0.88 KCNA5 (0.44) ITGB3ITGA2BF2TMPRSS6ITGAV
SCHEMBL7699209 0.88 F2 (0.42) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7415329 0.88 ITGB3 (0.35) ITGB3ITGA2BITGAVITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed