SCHEMBL7416019

SCHEMBL7416019

COc1ccccc1CN(C)CCN

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.71
CARM1 Q86X55 11/20 0.59
PRMT1 Q99873 11/20 0.59
TAAR1 Q96RJ0 1/20 0.58
MAOB P27338 3/20 0.57
AOC3 Q16853 1/20 0.56
BCHE P06276 2/20 0.55
ACHE P22303 2/20 0.55
CHRM1 P11229 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13706633 0.87 CHRM2 (0.82) CHRM2TAAR1MAOBBCHEACHE
SCHEMBL27909715 0.84 TAAR1 (0.59) CHRM2TAAR1MAOBAOC3BCHE
SCHEMBL19101439 0.84 CHRM2 (0.73) CHRM2MAOBAOC3BCHEACHE
SCHEMBL8705108 0.83 CHRM2 (0.71) CHRM2MAOBAOC3BCHEACHE
SCHEMBL4514454 0.80 CHRM2 (0.67) CHRM2TAAR1MAOBAOC3BCHE
SCHEMBL1133192 0.80 ACHE (0.55) CHRM2TAAR1MAOBAOC3BCHE
SCHEMBL4367373 0.80 ACHE (0.65) TAAR1MAOBBCHEACHE
SCHEMBL19080598 0.78 CHRM2 (0.72) CHRM2CARM1PRMT1MAOBBCHE
SCHEMBL735118 0.77 SLC6A4 (0.68) CHRM2TAAR1AOC3CHRM1
SCHEMBL11455232 0.77 CARM1 (0.58) CHRM2CARM1PRMT1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610165-A N-acylpiperidine tachykinin antagonists MERCK & CO., INC. (US) 1997-03-11 US disclosed
WO-1995022525-A1 N-ACYLPIPERIDINE TACHYKININ ANTAGONISTS MERCK & CO., INC. (US) 1995-08-24 WO disclosed
US-5344830-A Anitinflammatory, cardiovascular, analgesic, central nervous system MERCK & CO., INC. (US) 1994-09-06 US disclosed
WO-1994013646-A1 N,N-DIACYLPIPERAZINE TACHYKININ ANTAGONISTS MERCK & CO., INC. (US) 1994-06-23 WO disclosed