SCHEMBL7416111

SCHEMBL7416111

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)Cc2ccccc2[N+](=O)[O-])C(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.54
ITGA2B P08514 14/20 0.54
KDM4A O75164 1/20 0.51
PPARG P37231 3/20 0.40
ITGAV P06756 1/20 0.39
CHRM2 P08172 1/20 0.39
SLC6A4 P31645 1/20 0.39
MMP2 P08253 1/20 0.39
MMP9 P14780 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
KCNA5 P22460 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7418353 0.96 ITGB3 (0.51) ITGB3ITGA2BKDM4APPARGITGAV
SCHEMBL7418356 0.88 ITGB3 (0.41) ITGB3ITGA2BKDM4APPARG
SCHEMBL7698475 0.87 ITGB3 (0.50) ITGB3ITGA2BKDM4APPARGMMP2
Trifluoroacetic Acid SCHEMBL7415034 0.84 ITGB3 (0.47) ITGB3ITGA2BKDM4APPARGPPARA
SCHEMBL7412949 0.81 ITGB3 (0.55) ITGB3ITGA2BPPARGMMP2MMP9
SCHEMBL7409585 0.80 ITGB3 (0.61) ITGB3ITGA2BITGAVMMP2MMP9
SCHEMBL7411794 0.80 POLB (0.48) ITGB3ITGA2BMMP2MMP9KCNA5
SCHEMBL7695355 0.80 BCL2 (0.49) ITGB3ITGA2B
SCHEMBL7409554 0.80 MMP2 (0.61) ITGB3ITGA2BMMP2MMP9
SCHEMBL7463648 0.80 MAPT (0.46) ITGB3ITGA2BKDM4AMMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US claimed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP claimed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO claimed