SCHEMBL7418356

SCHEMBL7418356

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)Cc2ccccc2[N+](=O)[O-])C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.41
ITGA2B P08514 6/20 0.41
KDM4A O75164 1/20 0.40
F2 P00734 2/20 0.34
TMPRSS6 Q8IU80 2/20 0.34
BCL2 P10415 6/20 0.33
MCL1 Q07820 1/20 0.33
PPARG P37231 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7418353 0.90 ITGB3 (0.51) ITGB3ITGA2BKDM4AF2TMPRSS6
SCHEMBL7415041 0.89 AR (0.38) ITGB3ITGA2BKDM4AF2TMPRSS6
SCHEMBL7416111 0.88 ITGB3 (0.54) ITGB3ITGA2BKDM4APPARG
SCHEMBL7414953 0.83 ITGB3 (0.43) ITGB3ITGA2BF2TMPRSS6PPARG
SCHEMBL7420503 0.82 BCL2 (0.38) ITGB3ITGA2BF2TMPRSS6BCL2
SCHEMBL7414962 0.82 BCL2 (0.44) BCL2MCL1
SCHEMBL7417592 0.82 ITGB3 (0.49) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7423552 0.82 MAPT (0.41) ITGB3ITGA2BF2TMPRSS6BCL2
SCHEMBL7412096 0.81 MEN1 (0.43) ITGB3ITGA2BF2TMPRSS6
SCHEMBL7408399 0.81 F2 (0.47) ITGB3ITGA2BF2TMPRSS6PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed