SCHEMBL7416780

SCHEMBL7416780

CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(C(N)=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.54
CTSK P43235 1/20 0.54
CA2 P00918 1/20 0.52
MAPT P10636 2/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
GAA P10253 1/20 0.47
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 3/20 0.46
HSD17B10 Q99714 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HDAC4 P56524 2/20 0.45
HDAC1 Q13547 2/20 0.45
HPGD P15428 2/20 0.44
LMNA P02545 1/20 0.44
THRB P10828 1/20 0.44
KLK5 Q9Y337 1/20 0.44
EPHX2 P34913 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7407818 0.89 CTSS (0.54) CTSSCTSKCA2MAPTMEN1
SCHEMBL21585121 0.89 CTSS (0.54) CTSSCTSKCA2MAPTMEN1
SCHEMBL6555098 0.86 CTSS (0.56) CTSSCTSKCA2MAPTMEN1
SCHEMBL31075491 0.86 CTSS (0.56) CTSSCTSKCA2MAPTMEN1
SCHEMBL6557192 0.86 CTSS (0.56) CTSSCTSKCA2MAPTMEN1
SCHEMBL23975809 0.86 CTSS (0.61) CTSSCTSKCA2MAPTKDM4E
SCHEMBL7414151 0.86 CTSS (0.61) CTSSCTSKCA2MAPTKDM4E
SCHEMBL7414154 0.86 CTSS (0.61) CTSSCTSKCA2MAPTKDM4E
SCHEMBL21585117 0.85 CA2 (0.56) CTSSCTSKCA2MAPTMEN1
SCHEMBL21585118 0.84 CA2 (0.55) CTSSCTSKCA2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0796245-B1 PROCESS FOR THE PREPARATION OF AMIDINO PHENYL PYRROLIDINE BETA-ALANINE UREA ANALOGS SEARLE & CO (US) 2000-07-26 EP disclosed
US-5659063-A AMINE-BLOCKED METHIONINE ANALOG CYCLIZABLE TO A LACTAM IN NONVOLATILE OR NONTOXIC REAGENTS; ANTITHROMBOTIC AGENTS G. D. SEARLE & CO. (US) 1997-08-19 US disclosed
US-5610296-A CHEMICAL INTERMEDIATES OF ANTITHROMBOTICS G. D. SEARLE & CO. (US) 1997-03-11 US disclosed
US-5576447-A Process for the preparation of amidino phenyl pyrrolidine β-alanine urea analogs G. D. SEARLE & CO. (US) 1996-11-19 US disclosed
WO-1996017827-A1 PROCESS FOR THE PREPARATION OF AMIDINO PHENYL PYRROLIDINE β-ALANINE UREA ANALOGS G.D. SEARLE & CO. (US) 1996-06-13 WO disclosed
US-5484946-A CYCLIZATION AND DEHYDRATION A METHIONINE DERIVATIVE G. D. SEARLE & CO. (US) 1996-01-16 US disclosed