SCHEMBL741679

SCHEMBL741679

COCCCn1c(C2CCCN(C(=O)OC(C)(C)C)C2)nc2ccc(Cl)cc21

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV3 Q8NET8 1/20 0.41
ANO1 Q5XXA6 2/20 0.40
CNR1 P21554 3/20 0.40
CNR2 P34972 1/20 0.40
GLP1R P43220 1/20 0.39
KCNH2 Q12809 3/20 0.39
HRH1 P35367 2/20 0.39
CYP2D6 P10635 1/20 0.39
SCN9A Q15858 1/20 0.39
BRD4 O60885 1/20 0.39
USP30 Q70CQ3 1/20 0.39
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
HPGDS O60760 1/20 0.38
CHEK2 O96017 1/20 0.38
CHRM1 P11229 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741680 1.00 TRPV3 (0.41) TRPV3ANO1CNR1CNR2GLP1R
SCHEMBL762594 0.90 TRPV3 (0.43) TRPV3KCNH2HRH1CYP2D6SCN9A
SCHEMBL742014 0.90 HTT (0.43) KCNH2HRH1CYP2D6CHEK2CHRM1
SCHEMBL742013 0.90 HTT (0.43) KCNH2HRH1CYP2D6CHEK2CHRM1
SCHEMBL739667 0.89 KCNH2 (0.43) GLP1RKCNH2HRH1CYP2D6BRD4
SCHEMBL740873 0.88 SCN9A (0.45) TRPV3KCNH2HRH1CYP2D6SCN9A
SCHEMBL741974 0.88 KCNH2 (0.52) KCNH2HRH1CYP2D6HPGDSCHRM1
SCHEMBL741975 0.88 KCNH2 (0.52) KCNH2HRH1CYP2D6HPGDSCHRM1
SCHEMBL743901 0.88 ADORA2A (0.48) KCNH2HRH1CYP2D6CHEK2CHRM1
SCHEMBL743900 0.88 ADORA2A (0.48) KCNH2HRH1CYP2D6CHEK2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed