SCHEMBL740873

SCHEMBL740873

COCCCn1c(C2CCCN(C(=O)OC(C)(C)C)C2)nc2ccc(C(=O)OC)cc21

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.45
ADORA2A P29274 1/20 0.43
MC4R P32245 3/20 0.41
USP30 Q70CQ3 1/20 0.41
CHEK2 O96017 2/20 0.40
TRPV3 Q8NET8 1/20 0.40
MAPT P10636 2/20 0.39
TP53 P04637 1/20 0.39
THRB P10828 1/20 0.39
HPGDS O60760 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
KCNH2 Q12809 2/20 0.38
CYP2D6 P10635 1/20 0.38
HRH1 P35367 1/20 0.38
SYK P43405 1/20 0.38
ACSS2 Q9NR19 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762594 0.88 TRPV3 (0.43) SCN9ATRPV3MAPTTP53HPGDS
SCHEMBL741679 0.88 TRPV3 (0.41) SCN9AUSP30CHEK2TRPV3HPGDS
SCHEMBL741680 0.88 TRPV3 (0.41) SCN9AUSP30CHEK2TRPV3HPGDS
SCHEMBL742013 0.88 HTT (0.43) CHEK2MAPTKCNH2CYP2D6HRH1
SCHEMBL742014 0.88 HTT (0.43) CHEK2MAPTKCNH2CYP2D6HRH1
SCHEMBL741974 0.86 KCNH2 (0.52) HPGDSKCNH2CYP2D6HRH1
SCHEMBL741975 0.86 KCNH2 (0.52) HPGDSKCNH2CYP2D6HRH1
SCHEMBL743901 0.86 ADORA2A (0.48) ADORA2ACHEK2MAPTKCNH2CYP2D6
SCHEMBL743900 0.86 ADORA2A (0.48) ADORA2ACHEK2MAPTKCNH2CYP2D6
SCHEMBL740324 0.84 CYP2C9 (0.44) SCN9AUSP30TRPV3HPGDSKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed