SCHEMBL741975

SCHEMBL741975

COCCCn1c([C@@H]2CCCN(C(=O)OC(C)(C)C)C2)nc2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.52
HRH1 P35367 11/20 0.51
CYP2D6 P10635 6/20 0.51
CHRM1 P11229 3/20 0.51
USP2 O75604 1/20 0.47
POLB P06746 1/20 0.47
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
RXRG P48443 1/20 0.44
HPGDS O60760 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741974 1.00 KCNH2 (0.52) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL762625 0.89 CYP2C9 (0.44) KCNH2HRH1CYP2D6CHRM1HPGDS
SCHEMBL740324 0.89 CYP2C9 (0.44) KCNH2HRH1CYP2D6CHRM1HPGDS
SCHEMBL765031 0.89 P2RX3 (0.45) KCNH2HRH1CYP2D6CHRM1HPGDS
SCHEMBL741680 0.88 TRPV3 (0.41) KCNH2HRH1CYP2D6CHRM1HPGDS
SCHEMBL740716 0.88 CYP2D6 (0.41) KCNH2HRH1CYP2D6CHRM1HPGDS
SCHEMBL742013 0.88 HTT (0.43) KCNH2HRH1CYP2D6CHRM1
SCHEMBL762594 0.88 TRPV3 (0.43) KCNH2HRH1CYP2D6CHRM1HPGDS
SCHEMBL742014 0.88 HTT (0.43) KCNH2HRH1CYP2D6CHRM1
SCHEMBL741679 0.88 TRPV3 (0.41) KCNH2HRH1CYP2D6CHRM1HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed