SCHEMBL7417490

SCHEMBL7417490

O=C(CCl)c1ccc2c(c1)C1(CCCC1)C(=O)N2

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PGR P06401 7/20 0.50
IP6K1 Q92551 8/20 0.49
IP6K3 Q96PC2 1/20 0.49
IP6K2 Q9UHH9 1/20 0.49
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
MAPK14 Q16539 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20268055 0.83 PGR (0.47) PGRIP6K1IP6K3IP6K2PDE4A
SCHEMBL9773678 0.82 IP6K1 (0.63) PGRIP6K1IP6K3IP6K2PDE4A
SCHEMBL20268826 0.81 IP6K1 (0.55) PGRIP6K1IP6K3IP6K2PDE4A
SCHEMBL10520525 0.80 IP6K1 (0.48) PGRIP6K1IP6K3IP6K2
SCHEMBL20268320 0.78 IP6K1 (0.55) PGRIP6K1IP6K3IP6K2PDE4A
SCHEMBL5680486 0.78 PGR (0.50) PGRALDH1A1MAPTPDE3BPDE3A
SCHEMBL12548325 0.77 IP6K1 (0.57) PGRIP6K1IP6K3IP6K2ALDH1A1
SCHEMBL16849906 0.77 IP6K1 (0.60) PGRIP6K1IP6K3IP6K2
SCHEMBL8524882 0.76 ALDH1A1 (0.47) ALDH1A1MAPT
SCHEMBL23590773 0.76 PGR (0.40) PGRPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281309-B1 PIPERAZINYL-HETEROCYCLIC COMPOUNDS PFIZER INC. (US) 1991-12-27 EP disclosed
US-4883795-A Piperazinyl-heterocyclic compounds PFIZER INC. (US) 1989-11-28 US disclosed
US-4831031-A Aryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activity PFIZER INC. (US) 1989-05-16 US disclosed