SCHEMBL7417577

SCHEMBL7417577

CN(C)C(C#N)c1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.47
CFTR P13569 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
GOPC Q9HD26 1/20 0.44
KCNA5 P22460 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1999341 0.82 CFTR (0.44) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL10664321 0.79 CYP19A1 (0.49) CYP19A1SMN1; SMN2KDM4E
SCHEMBL1275688 0.77 TRPA1 (0.46) SMN1; SMN2KDM4E
SCHEMBL3447644 0.77 TRPA1 (0.46) SMN1; SMN2KDM4E
SCHEMBL9314550 0.76 CYP19A1 (0.51) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL17591685 0.75 CFTR (0.52) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL7021489 0.75 CYP19A1 (0.55) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL27929742 0.74 OPRM1 (0.52) CFTRSLC6A2SLC6A4SLC6A3GOPC
Hydrochloric Acid SCHEMBL1477644 0.73 MEN1 (0.37) CFTRSLC6A2SLC6A4SLC6A3GOPC
SCHEMBL6581568 0.73 CFTR (0.50) CYP19A1CFTRSLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994373-A COGNITION ACTIVATORS; GASTROINTESTINAL DISORDERS; PSYCHOLOGICAL DISORDERS NOVO NORDISK A/S NOVO ALLE DK 2880 (DK) 1999-11-30 US disclosed
EP-0835255-A1 NOVEL SUBSTITUTED AZACYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1998-04-15 EP disclosed
WO-1997001555-A1 NOVEL SUBSTITUTED AZACYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1997-01-16 WO disclosed