SCHEMBL7417679

SCHEMBL7417679

COC(=O)C(CC(=O)O)NC(=O)c1ccc(-c2ccccc2S(=O)(=O)NC(C)C)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.51
USP30 Q70CQ3 1/20 0.47
OPRM1 P35372 1/20 0.47
OPRK1 P41145 1/20 0.47
CYP26A1 O43174 1/20 0.43
POLB P06746 1/20 0.42
GAA P10253 2/20 0.41
RAB9A P51151 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP2C9 P11712 1/20 0.41
ALOX12 P18054 1/20 0.41
CYP2C19 P33261 1/20 0.41
RECQL P46063 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
CYCS P99999 1/20 0.41
CA2 P00918 3/20 0.41
CA1 P00915 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
F10 P00742 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415012 0.87 CYP26A1 (0.46) CASP1CYP26A1GAARAB9AALDH1A1
SCHEMBL7417684 0.86 CASP1 (0.44) CASP1CYP26A1GAARAB9AGPR55
SCHEMBL7423070 0.77 USP30 (0.49) USP30GAARAB9ACA2CA1
SCHEMBL23967346 0.77 GAA (0.54) CASP1CYP26A1GAARAB9AALDH1A1
SCHEMBL7464416 0.76 CA1 (0.47) CYP26A1GAARAB9AALDH1A1SMN1; SMN2
SCHEMBL5191776 0.76 OPRM1 (0.63) CASP1OPRM1OPRK1ALDH1A1SMN1; SMN2
SCHEMBL1109199 0.69 CYP26A1 (0.59) CYP26A1GAARAB9AALDH1A1SMN1; SMN2
SCHEMBL29067682 0.68 GAA (0.53) CYP26A1POLBGAARAB9AALDH1A1
SCHEMBL13868571 0.68 GAA (0.53) CYP26A1POLBGAARAB9AALDH1A1
SCHEMBL4896289 0.68 GAA (0.53) CYP26A1POLBGAARAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235807-A1 B-AMINO ACID-, ASPARTIC ACID- AND DIAMINOPROPIONIC-BASED INHIBITORS OF FACTOR XA Millennium Pharmaceuticals, Inc. (US) 2002-09-04 EP disclosed
WO-2001038309-A1 β-AMINO ACID-, ASPARTIC ACID- AND DIAMINOPROPIONIC-BASED INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2001-05-31 WO disclosed