SCHEMBL7464416

SCHEMBL7464416

COC(=O)C(CC(=O)OCc1ccccc1)NC(=O)c1ccc(-c2ccccc2S(C)(=O)=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
F10 P00742 4/20 0.46
PRSS1 P07477 1/20 0.46
RAB9A P51151 2/20 0.44
MAPT P10636 2/20 0.44
GAA P10253 1/20 0.44
CYP26A1 O43174 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TP53 P04637 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MMP9 P14780 1/20 0.40
KYNU Q16719 1/20 0.39
LMNA P02545 1/20 0.39
GLA P06280 1/20 0.39
ACE P12821 1/20 0.39
CTSB P07858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423070 0.89 USP30 (0.49) CA1CA2F10PRSS1RAB9A
SCHEMBL7415012 0.88 CYP26A1 (0.46) CA1CA2F10RAB9AGAA
SCHEMBL3540630 0.78 RAB9A (0.54) RAB9AMAPTGAACYP26A1MEN1
SCHEMBL3534617 0.77 MEN1 (0.54) CA1CA2RAB9AMAPTMEN1
SCHEMBL7417679 0.76 CASP1 (0.51) CA1CA2F10RAB9AGAA
SCHEMBL7418216 0.75 F10 (0.56) F10RAB9AMAPTGAAMEN1
SCHEMBL7417684 0.74 CASP1 (0.44) CA1CA2F10PRSS1RAB9A
Trifluoroacetic Acid SCHEMBL6165833 0.74 F10 (0.58) F10PRSS1
SCHEMBL16667936 0.74 GAA (0.58) RAB9AGAAALDH1A1MMP9LMNA
Trifluoroacetic Acid SCHEMBL6165839 0.73 ALDH1A1 (0.44) CA1CA2F10PRSS1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235807-A1 B-AMINO ACID-, ASPARTIC ACID- AND DIAMINOPROPIONIC-BASED INHIBITORS OF FACTOR XA Millennium Pharmaceuticals, Inc. (US) 2002-09-04 EP disclosed
WO-2001038309-A1 β-AMINO ACID-, ASPARTIC ACID- AND DIAMINOPROPIONIC-BASED INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2001-05-31 WO disclosed