SCHEMBL7417787

SCHEMBL7417787

Cc1cccc2[nH]c(N3CCCN(C(C)C)CC3)nc12

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.47
AURKA O14965 1/20 0.43
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
PARP1 P09874 8/20 0.40
HRH4 Q9H3N8 1/20 0.39
OGA O60502 1/20 0.38
ALKBH3 Q96Q83 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
GAA P10253 4/20 0.37
MGAM O43451 3/20 0.37
SI P14410 3/20 0.37
MGAM2 Q2M2H8 3/20 0.37
KDM4E B2RXH2 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5620810 0.82 PARP1 (0.64) PARP1PARP2
SCHEMBL7759238 0.82 MGAM (0.51) AURKAACHEPARP1PARP2GAA
SCHEMBL11198421 0.80 HRH4 (0.58) NPY5RAURKAPARP1HRH4ALKBH3
SCHEMBL6864586 0.79 PARP1 (0.45) NPY5RPARP1PARP2
SCHEMBL7411395 0.77 NPY5R (0.45) NPY5RAURKABCHEACHEPARP1
SCHEMBL7600366 0.77 HTR3A (0.59) NPY5RAURKABCHEACHEPARP1
SCHEMBL7762915 0.76 MGAM (0.55) AURKAACHEPARP1PARP2GAA
SCHEMBL5620966 0.76 PARP1 (0.69) PARP1PARP2
SCHEMBL7417491 0.74 NPY5R (0.45) NPY5RPARP1PARP2
SCHEMBL6869126 0.73 PARP1 (0.48) NPY5RPARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed