SCHEMBL7600366

SCHEMBL7600366

Cc1cccc2[nH]c(N3CCNCC3)nc12

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 2/20 0.59
NPY5R Q15761 1/20 0.54
AURKA O14965 1/20 0.50
ADRB1 P08588 2/20 0.47
HTR6 P50406 2/20 0.47
HRH4 Q9H3N8 1/20 0.45
PIM1 P11309 1/20 0.44
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
MGAM O43451 4/20 0.43
GAA P10253 4/20 0.43
SI P14410 4/20 0.43
MGAM2 Q2M2H8 4/20 0.43
ALKBH3 Q96Q83 1/20 0.43
PARP1 P09874 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11198421 0.85 HRH4 (0.58) HTR3ANPY5RAURKAHTR6HRH4
SCHEMBL20449682 0.77 PARP1 (0.56) HTR3AHTR6PARP1
SCHEMBL17697629 0.77 CRBN (0.59) HTR3AHTR6PARP1
SCHEMBL7417787 0.77 NPY5R (0.47) NPY5RAURKAHRH4MGAMGAA
SCHEMBL1066810 0.76 HTR3A (0.56) HTR3ANPY5RADRB1HTR6PIM1
SCHEMBL5621808 0.76 PARP1 (0.72) PARP1
SCHEMBL28034227 0.75 HTR3A (0.51) HTR3ANPY5RHTR6PIM1PARP1
SCHEMBL28034117 0.75 HTR3A (0.48) HTR3ANPY5RHTR6PIM1PARP1
SCHEMBL5506042 0.75 HTR3A (0.48) HTR3ANPY5RHTR6HRH4PIM1
SCHEMBL7463681 0.74 ADRB1 (0.44) HTR3AADRB1HRH4PIM1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255736-A2 SUBSTITUTED PIPERAZINE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) Boehringer Ingelheim Pharma KG (DE) 2002-11-13 EP disclosed
WO-2001047898-A2 SUBSTITUTED PIPERAZINE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-07-05 WO disclosed