SCHEMBL741786

SCHEMBL741786

COCCCNc1cccc(OC)c1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.49
HPGD P15428 2/20 0.46
MAPT P10636 2/20 0.46
HSD17B10 Q99714 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HTT P42858 1/20 0.44
HTR1A P08908 2/20 0.43
ADRA1D P25100 2/20 0.43
ADRA1A P35348 2/20 0.43
ADRA1B P35368 2/20 0.43
PTGER4 P35408 1/20 0.41
KDM4E B2RXH2 2/20 0.40
GAA P10253 2/20 0.40
ALDH1A1 P00352 1/20 0.40
KCNH3 Q9ULD8 1/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2219253 0.95 CHRM2 (0.51) CHRM2HPGDMAPTHSD17B10SMN1; SMN2
SCHEMBL20837291 0.90 NCF1 (0.44) CHRM2HPGDMAPTHSD17B10SMN1; SMN2
SCHEMBL2476416 0.81 KDM4E (0.47) CHRM2MAPTHSD17B10HTTHTR1A
SCHEMBL20232562 0.78 ALDH1A1 (0.42) CHRM2HPGDMAPTHSD17B10SMN1; SMN2
SCHEMBL2217667 0.77 HTT (0.40) CHRM2HPGDMAPTHSD17B10SMN1; SMN2
SCHEMBL7745287 0.77 PTGER4 (0.51) CHRM2HPGDMAPTHSD17B10SMN1; SMN2
SCHEMBL739875 0.77 MAPT (0.58) CHRM2HPGDMAPTSMN1; SMN2HTT
Sulfuric Acid SCHEMBL7104162 0.75 KDM4E (0.46) CHRM2HSD17B10HTTHTR1AADRA1D
SCHEMBL7771127 0.73 CHRM2 (0.62) CHRM2MAPTHSD17B10KDM4EGAA
SCHEMBL1421223 0.73 MAPT (0.54) CHRM2HPGDMAPTHTTHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed