SCHEMBL7418261

SCHEMBL7418261

COc1ccc(Br)c(C(=O)N[C@@H](Cc2ccc(-c3c(C)c(Br)c[nH]c3=O)cc2)C(=O)O)c1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 10/20 0.61
ITGB1 P05556 9/20 0.61
ITGB2 P05107 2/20 0.56
ICAM1 P05362 2/20 0.56
ITGAL P20701 2/20 0.56
PIN1 Q13526 1/20 0.45
CA2 P00918 1/20 0.43
ITGB7 P26010 7/20 0.42
ALB P02768 1/20 0.41
IL2 P60568 1/20 0.41
HPGD P15428 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ALOX15 P16050 1/20 0.39
PTPN1 P18031 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414372 0.93 ITGB1 (0.52) ITGA4ITGB1ITGB2ICAM1ITGAL
SCHEMBL7415187 0.88 ITGB1 (0.61) ITGA4ITGB1ITGB2ICAM1ITGAL
SCHEMBL7416080 0.81 ITGB1 (0.52) ITGA4ITGB1ITGB2ICAM1ITGAL
SCHEMBL4649073 0.78 ITGA4 (0.59) ITGA4ITGB1ITGB2ICAM1ITGAL
SCHEMBL4649064 0.78 ITGA4 (0.59) ITGA4ITGB1ITGB2ICAM1ITGAL
SCHEMBL4893859 0.75 ITGA4 (0.78) ITGA4ITGB1ITGB2ICAM1ITGAL
SCHEMBL4892883 0.75 ITGA4 (1.00) ITGA4ITGB1ITGB2ICAM1ITGAL
SCHEMBL5162599 0.75 ITGA4 (0.74) ITGA4ITGB1ITGB2ICAM1ITGAL
SCHEMBL5133478 0.73 ITGA4 (0.79) ITGA4ITGB1ITGB2ICAM1ITGAL
SCHEMBL4648129 0.72 ITGA4 (0.53) ITGA4ITGB1ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244625-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-10-02 EP claimed
WO-2001042215-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO claimed
EP-1244625-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-10-02 EP disclosed
WO-2001042215-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed