SCHEMBL7416080

SCHEMBL7416080

COC(=O)[C@H](Cc1ccc(-c2c(C)cc[nH]c2=O)cc1)NC(=O)c1cc(OC)ccc1Br

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.52
ITGA4 P13612 2/20 0.52
ITGB2 P05107 1/20 0.45
ICAM1 P05362 1/20 0.45
ITGAL P20701 1/20 0.45
HPGD P15428 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
PKM P14618 1/20 0.40
KDR P35968 1/20 0.38
PIN1 Q13526 2/20 0.38
HDAC1 Q13547 6/20 0.38
HDAC6 Q9UBN7 6/20 0.38
LNPEP Q9UIQ6 1/20 0.38
TACR3 P29371 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415187 0.93 ITGB1 (0.61) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL7414372 0.88 ITGB1 (0.52) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL7418261 0.81 ITGA4 (0.61) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL7418253 0.76 ITGB1 (0.57) ITGB1ITGA4
SCHEMBL7422329 0.76 ITGA4 (0.48) ITGA4
SCHEMBL6240483 0.75 ITGA4 (0.87) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL6239694 0.75 ITGB1 (0.68) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL4648805 0.74 ITGB1 (0.49) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL4648806 0.74 ITGB1 (0.49) ITGB1ITGA4ITGB2ICAM1ITGAL
Hydrochloric Acid SCHEMBL7419313 0.72 ALDH1A1 (0.42) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244625-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-10-02 EP disclosed
WO-2001042215-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed