SCHEMBL7419102

SCHEMBL7419102

OCc1cccc(-c2ncc[nH]2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.42
MTOR P42345 1/20 0.42
ADK P55263 1/20 0.42
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADRA2A P08913 2/20 0.36
CSNK1A1 P48729 1/20 0.36
TYRO3 Q06418 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
KDM4E B2RXH2 2/20 0.36
CBFB Q13951 2/20 0.35
NUDT1 P36639 1/20 0.35
PARP1 P09874 1/20 0.35
CCR1 P32246 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP19A1 P11511 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL197279 0.82 NISCH (0.54) NISCHMTORADKALDH1A1MEN1
SCHEMBL13830975 0.78 NISCH (0.39) NISCHMTORADKALDH1A1MEN1
SCHEMBL28596107 0.76 ALDH1A1 (0.38) NISCHMTORADKALDH1A1MEN1
SCHEMBL16588099 0.75 CCR1 (0.48) ALDH1A1MEN1KMT2AKDM4ECCR1
SCHEMBL29079328 0.75 NISCH (0.47) NISCHMTORADKALDH1A1MEN1
SCHEMBL14304159 0.74 NISCH (0.46) NISCHMTORADKALDH1A1MEN1
SCHEMBL309114 0.74 CCR1 (0.54) NISCHMTORADKALDH1A1MEN1
SCHEMBL4766313 0.74 NISCH (0.46) NISCHMTORADKALDH1A1MEN1
SCHEMBL31374443 0.74 NISCH (0.46) NISCHMTORADKALDH1A1MEN1
SCHEMBL3050014 0.74 NISCH (0.46) NISCHMTORADKALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113121502-A Heteroaromatic hydrocarbon compound, intermediate, composition and application 山东铂源生物医药有限公司 2021-07-16 CN disclosed
EP-0986562-A1 SUBSTITUTED 1,2,4-TRIAZOLO 3,4-A]PHTHALAZINE DERIVATIVES AS GABA ALPHA 5 LIGANDS MERCK SHARP & DOHME LTD. (GB) 2000-03-22 EP disclosed
WO-1998050385-A1 SUBSTITUTED 1,2,4-TRIAZOLO[3,4-a]PHTHALAZINE DERIVATIVES AS GABA ALPHA 5 LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1998-11-12 WO disclosed