SCHEMBL741940

SCHEMBL741940

CC1(C)OC2CC(N)C(N)(C(=O)c3cc4cc(Cl)ccc4[nH]3)CC2O1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.43
F7 P08709 1/20 0.43
F3 P13726 1/20 0.43
FLT3 P36888 1/20 0.42
HRH4 Q9H3N8 9/20 0.41
HRH3 Q9Y5N1 5/20 0.41
HRH1 P35367 1/20 0.40
PYGL P06737 5/20 0.40
MEN1 O00255 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
KMT2A Q03164 2/20 0.39
IDO1 P14902 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL743632 0.80 FLT3 (0.48) SMYD3F7F3FLT3HRH4
SCHEMBL743134 0.79 FLT3 (0.47) SMYD3F7F3FLT3HRH4
SCHEMBL11888291 0.77 HRH4 (0.47) SMYD3F7F3HRH4HRH3
SCHEMBL740522 0.77 SMYD3 (0.48) SMYD3F7F3FLT3HRH4
SCHEMBL764007 0.77 SMYD3 (0.56) SMYD3HRH4PYGL
SCHEMBL4083338 0.77 SMYD3 (0.56) SMYD3HRH4PYGL
SCHEMBL4087518 0.77 SMYD3 (0.56) SMYD3HRH4PYGL
SCHEMBL27520223 0.74 SMYD3 (0.45) SMYD3F7F3FLT3HRH4
SCHEMBL743889 0.74 HRH4 (0.46) SMYD3F7F3FLT3HRH4
SCHEMBL742510 0.74 F10 (0.65)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed
US-7935824-B2 Ethylenediamine derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2011-05-03 US disclosed